A protein family as ChEMBL classifies it.
servable in this model
measured here and in at least one other family
involving this family
| Quantity | Value |
|---|---|
| Measurements | 38 |
| Activity range, pActivity | 2.92 to 8.17 |
| Median activity | 5.07 |
| Endpoint | Measurements |
|---|---|
| Ki | 19 |
| IC50 | 15 |
| Kd | 3 |
| EC50 | 1 |
Every ligand counted here is measured in this family and in at least one other. The question worth asking is how many families a compound reaches altogether, because a compound seen in four families is a very different starting point from one seen in two.
| Families a compound reaches | Compounds |
|---|---|
| Two | 3 |
| Three | 1 |
| Four or more | 6 |
| Family | Shared compounds |
|---|---|
| Oxidoreductase | 5 |
| Electrochemical transporter | 5 |
| Nuclear receptor | 4 |
| Transferase | 4 |
| Primary active transporter | 4 |
| Lyase | 4 |